Granisetron hydrochloride

Catalog # Availability Size / Price Qty
Granisetron hydrochloride | CAS No. 107007-99-8 | 5-HT3 Receptor Antagonists
1 Image
Description: 5-HT3 antagonist
Alternative Names: BRL 43694

Chemical Name: 1-Methyl-N-[(3-endo)-9-methyl-9-azabicyclo[3.3.1]non-3-yl]-1H-indazole-3-carboxamide hydrochloride

Purity: ≥99%

Product Details
Citations (4)
Supplemental Products

Biological Activity

Granisetron hydrochloride is a 5-HT3 receptor antagonist that possesses potent antiemetic activity.

Technical Data

Soluble to 100 mM in water and to 10 mM in DMSO
Desiccate at +4°C

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Selective and functional 5-hydroxytryptamine3 receptor antagonism by BRL 43694 (granisetron).
    Sanger and Nelson
    Eur.J.Pharmacol., 1989;159:113
  2. Granisetron. A review of its pharmacological properties and therapeutic use as an antiemetic.
    Plosker and Goa
    Drugs, 1991;42:805
  3. Anti-emetic effect of ondans. and granis. after exposure to mixed neutron and gamma irradiation.
    Martin et al.
    Rad.Res., 1998;149:631

Product Datasheets

Or select another batch:
Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.


Molarity Calculator


*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

Citations for Granisetron hydrochloride

The citations listed below are publications that use Tocris products. Selected citations for Granisetron hydrochloride include:

4 Citations: Showing 1 - 4


No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs

Reviews for Granisetron hydrochloride

There are currently no reviews for this product. Be the first to review Granisetron hydrochloride and earn rewards!

Have you used Granisetron hydrochloride?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.