GRK2 inhibitory polypeptide that specifically inhibits Gβγ
activation of GRK2. Corresponds to the Gβγ
-binding domain and acts as a cellular Gβγ
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Cellular expression of the carboxyl terminus of a G protein-coupled receptor kinase attenuates Gβγ-mediated signaling.
Koch et al.
A βγ dimer derived from G13 transduces the angiotensin AT1 receptor signal to stimulation of Ca2+ channels in rat portal vein myocytes.
Macrez et al.
Two distinct mechanisms mediate acute μ-opioid receptor desensitization in native neurons.
Dang et al.
The citations listed below are publications that use Tocris products. Selected citations for GRK2i include:
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