HS 024

Catalog # Availability Size / Price Qty
1832/1
HS 024
1 Image
Description: Highly potent MC4 receptor antagonist
Product Details
Citations (2)
Supplemental Products
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Biological Activity

Highly potent melanocortin MC4 receptor antagonist (Ki values are 0.29, 18.6, 5.45 and 3.29 nM for cloned human MC4, MC1, MC3 and MC5 receptors respectively). Increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats, following central administration in vivo.

Technical Data

M.Wt:
1266.5
Formula:
C58H79N19O10S2
Sequence:
CXRHXRWGC

(Modifications: Cys-1 = N-terminal Ac, X-2 = Nle, X-5 = Nal, Cys-9 = C-terminal amide, Disulfide bridge between 1 - 9)

Solubility:
Soluble to 0.50 mg/ml in water
Storage:
Desiccate at -20°C
CAS No:
212370-59-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

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Citations for HS 024

The citations listed below are publications that use Tocris products. Selected citations for HS 024 include:

2 Citations: Showing 1 - 2

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