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JNJ 5207787

4018 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
4018/10
4018/50
JNJ 5207787 | CAS No. 683746-68-1 | NPY Receptor Antagonists
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Description: Selective NPY Y2 receptor antagonist

Chemical Name: (2E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cyanophenyl)-N-[1-(2-cyclopentylethyl)-4-piperidinyl]-2-propenamide

Purity: ≥98%

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Biological Activity

Selective NPY Y2 antagonist (IC50 = 0.1 μM). Displays 100-fold selectivity over NPY Y1, Y4 and Y5 receptors; also displays selectivity against a panel of 50 receptors, ion channels and transporters. Brain penetrant.

Technical Data

M.Wt:
510.67
Formula:
C32H38N4O2
Solubility:
Soluble to 10 mM in DMSO with gentle warming and to 10 mM in ethanol with gentle warming
Purity:
≥98%
Storage:
Store at RT
CAS No:
683746-68-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold with the permission of Janssen Pharmaceutica N.V.

Product Datasheets

Reconstitution Calculator
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Reconstitution Calculator

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VersaClone cDNA Plasmids

Human NPY2R (NP_000901) VersaClone cDNA

RDC0157

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