Home / NPY Receptor Antagonists / JNJ 5207787

JNJ 5207787

4018 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
4018/10
4018/50
NPY Receptor Antagonists Small Molecule
1 Image
Description: Selective NPY Y2 receptor antagonist

Chemical Name: (2E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cyanophenyl)-N-[1-(2-cyclopentylethyl)-4-piperidinyl]-2-propenamide

Purity: ≥98%

Product Details
Supplemental Products
Reviews
Biological Activity Technical Data Additional Information Background Product Datasheets Calculators

Biological Activity

Selective NPY Y2 antagonist (IC50 = 0.1 μM). Displays 100-fold selectivity over NPY Y1, Y4 and Y5 receptors; also displays selectivity against a panel of 50 receptors, ion channels and transporters. Brain penetrant.

Technical Data

M.Wt:
510.67
Formula:
C32H38N4O2
Solubility:
Soluble to 10 mM in DMSO with gentle warming and to 10 mM in ethanol with gentle warming
Purity:
≥98%
Storage:
Store at RT
CAS No:
683746-68-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold with the permission of Janssen Pharmaceutica N.V.

Product Datasheets

Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Molarity Calculator

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / CoA (available online).

FAQs

No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs

VersaClone cDNA Plasmids

Human NPY2R (NP_000901) VersaClone cDNA

RDC0157

Reviews for JNJ 5207787

There are currently no reviews for this product. Be the first to review JNJ 5207787 and earn rewards!

Have you used JNJ 5207787?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.