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Catalog Number:4018
Chemical Name:(2E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cyanophenyl)-N-[1-(2-cyclopentylethyl)-4-piperidinyl]-2-propenamide
Product Details
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Biological Activity
Selective NPY Y2 antagonist (IC50 = 0.1 μM). Displays 100-fold selectivity over NPY Y1, Y4 and Y5 receptors; also displays selectivity against a panel of 50 receptors, ion channels and transporters. Brain penetrant.
Selective NPY Y2 antagonist (IC50 = 0.1 μM). Displays 100-fold selectivity over NPY Y1, Y4 and Y5 receptors; also displays selectivity against a panel of 50 receptors, ion channels and transporters. Brain penetrant.
Technical Data
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M.Wt:510.67
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Formula:C32H38N4O2
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Solubility:Soluble to 10 mM in DMSO with gentle warming and to 10 mM in ethanol with gentle warming
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Purity:>98
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Storage:Store at RT
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CAS No:683746-68-1
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Additional Information
Licensing Caveats:
Sold with the permission of Janssen Pharmaceutica N.V.
Product Datasheets
Tocris Bioscience is the leading supplier of novel and exclusive tools for
life science research with over 30 years' experience in the industry.
Tocris is a Bio-Techne brand.