Selective inhibitor of the breast cancer resistance protein (BCRP) multidrug transporter (IC50
values are 0.59 and 1.39 μ
M in Pheo A and Hoechst 33342 assays respectively). Displays no inhibitory activity against P-gp or MRP1.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Specific inhibitors of the breast cancer resistance protein (BCRP).
Pick et al.