KW 3902

( 1 Review )    
Product Datasheet
Catalog Number:4167
Alternate Names:Rolofylline
Chemical Name:8-(Hexahydro-2,5-methanopentalen-3a(1H)-yl)-3,7-dihydro-1,3-dipropyl-1H-purine-2,6-dione
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Biological Activity
Selective adenosine A1 receptor antagonist; displays 890-fold selectivity for rat A1 receptors over A2A receptors (Ki values are 0.19 and 170 nM respectively). Displays no effect on recombinant rat A3 receptors expressed on CHO cells at concentrations up to 10 μM. Exhibits diuretic and renal protective effects in rats.
Technical Data
  • M.Wt:
    356.46
  • Formula:
    C20H28N4O2
  • Solubility:
    Soluble to 50 mM in DMSO and to 25 mM in ethanol
  • Purity:
    >99
  • Storage:
    Store at +4°C
  • CAS No:
    136199-02-5
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
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VersaClone cDNA Plasmids
Description Application Cat# Citations Images  

Human Adenosine A1 R (NP_000665) VersaClone cDNA

RDC0213
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Mouse Adenosine A1 R (NP_000665) VersaClone cDNA

RDC2041
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Average Rating: 5 (Based on 1 review)

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  Mouse Ariel Vitenzon 01/05/2018
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Summary

Species Mouse

Other Experimental Details

Other Experimental Details The drug dissolves well in saline + 0.3% tween 80 with 3X vortex (1min) and sonicate (5min).

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Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.

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