Selective cholecystokinin receptor 2 (CCK2
) antagonist (IC50
values are 2 and 280 nM at CCK2
receptors respectively) that is inactive at a range of other receptors including opiate, muscarinic acetylcholine, α
- and β
adrenergic, histamine, angiotensin and bradykinin receptors.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Cholecystokinin action on layer 6b neurons in somatosensory cortex.
Chung et al.
Brain Res., 2009;1282:10
Benzodiazepine gastrin and brain cholecystokinin receptor ligands: L-365,260.
Kees et al.
A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-B) ligand: L-365,260.
Lotti and Chang
The citations listed below are publications that use Tocris products. Selected citations for L-365,260 include:
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