Biological Activity Potent, non-peptide and orally active oxytocin receptor antagonist (IC50 = 8.9 nM) that displays > 40-fold selectivity over vasopressin V1a and V2 receptors (IC50 values are 370 and 570 nM respectively). Antagonizes oxytocin-induced uterine contractions in vitro and in vivo.
Soluble to 100 mM in water and to 100 mM in DMSO
Store at -20°C
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For batch specific data refer to the Certificate of Analysis.
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