Leelamine hydrochloride

Tocris Bioscience | Catalog # 2139

CB1 agonist
Tocris Bioscience
Discontinued Product
2139 has been discontinued. View all Cannabinoid R1/CB1 Agonists products.

Key Product Details

Description

CB1 agonist

Alternative Names

Lylamine hydrochloride,(+)-Dehydroabietylamine
View all Cannabinoid R1/CB1 Agonists »

Product Description

Leelamine hydrochloride is a CB1 agonist. Displaces binding of [3H]-SR141716A with an IC50 value of 2.86 μM.

Product Specifications for Leelamine hydrochloride

Molecular Weight

321.93

Formula

C20H31N.HCl

Storage

Store at -20°C

Purity

≥98% (HPLC)

Chemical Name

(1R,4aS,10aR)-1,2,3,4,4a,9,10,10a-Octahydro-1-,4a-dimethyl-7-(1-methylethyl)-1-phenanthrenemethanamine hydrochloride

CAS Number

16496-99-4

PubChem ID

16759156

InChI Key

CVPQLGCAWUAYPF-WFBUOHSLSA-N

SMILES

NC[C@]1(C)CCC[C@@]3(C)[C@]([H])1CCC2=CC(C(C)C)=CC=C23.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 32.19 100
Ethanol 32.19 100

Preparing Stock Solutions for Leelamine hydrochloride

The following data is based on the product molecular weight 321.93.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 3.11 mL 15.53 mL 31.06 mL
5 mM 0.62 mL 3.11 mL 6.21 mL
10 mM 0.31 mL 1.55 mL 3.11 mL
50 mM 0.06 mL 0.31 mL 0.62 mL

Calculators

Calculate the mass, volume, or concentration required for a solution.

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

Calculate the dilution required to prepare a stock solution.

x
=
x

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 19 publications citing the usage of this product.

There are currently no references for this product.

Product Documents for Leelamine hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Leelamine hydrochloride

For research use only

Related Research Areas

Bioactive Lipids and Receptors

Citations for Leelamine hydrochloride

Customer Reviews for Leelamine hydrochloride

There are currently no reviews for this product. Be the first to review Leelamine hydrochloride and earn rewards!

Have you used Leelamine hydrochloride?

Submit a review and receive an Amazon gift card!

$25/€18/£15/$25CAN/¥2500 Yen for a review with an image

$10/€7/£6/$10CAN/¥1110 Yen for a review without an image

Submit a review
Amazon Gift Card