LY 255283

Catalog # Availability Size / Price Qty
2208/10
2208/50
LY 255283 | CAS No. 117690-79-6 | Leukotriene and Related Receptor Antagonists
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Description: Selective, competitive BLT2 receptor antagonist

Chemical Name: 1-[5-Ethyl-2-hydroxy-4-[[6-methyl-6-(1H-tetrazol-5-yl)heptyl]oxy]phenyl]ethanone

Purity: ≥98%

Product Details
Citations (1)
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Biological Activity

Selective, competitive antagonist of BLT2 receptors (IC50 values are ~ 1 and > 10 μM at human recombinant BLT2 and BLT1 receptors respectively). Inhibits LTB4-induced contraction of lung parenchyma (pA2 = 7.2), and reduces LTB4-mediated airway obstruction in guinea pigs following i.v. and oral administration..

Technical Data

M.Wt:
360.46
Formula:
C19H28N4O3
Solubility:
Soluble to 100 mM in DMSO and to 25 mM in ethanol
Purity:
≥98%
Storage:
Store at +4°C
CAS No:
117690-79-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citation for LY 255283

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