LY 266097 hydrochloride

Tocris Bioscience | Catalog # 4081

Selective 5-HT2B antagonist
Tocris Bioscience

Key Product Details

Description

Selective 5-HT2B antagonist
View all 5-HT2B Receptor Antagonists »

Product Description

LY 266097 hydrochloride is a selective 5-HT2B receptor antagonist (pKi = 9.3). More than 100-fold selective over 5-HT2A and 5-HT2C. Attenuates amphetamine-induced locomotion in the rat.

Product Specifications for LY 266097 hydrochloride

Molecular Weight

407.33

Formula

C21H23ClN2O2.HCl

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

1-[(2-Chloro-3,4-dimethoxyphenyl)methyl]-2,3,4,9-tetrahydro-6-methyl-1H-pyrido[3,4-b]indole hydrochloride

CAS Number

172895-39-5

PubChem ID

9953184

InChI Key

KPXKZZURYAXZQE-UHFFFAOYSA-N

SMILES

CC1=CC=C(NC3=C2CCNC3CC4=CC=C(OC)C(OC)=C4Cl)C2=C1.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 40.73 100
Ethanol 40.73 100

Preparing Stock Solutions for LY 266097 hydrochloride

The following data is based on the product molecular weight 407.33.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.46 mL 12.28 mL 24.55 mL
5 mM 0.49 mL 2.46 mL 4.91 mL
10 mM 0.25 mL 1.23 mL 2.46 mL
50 mM 0.05 mL 0.25 mL 0.49 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 3 publications citing the usage of this product.

Product Documents for LY 266097 hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for LY 266097 hydrochloride

For research use only

Citations for LY 266097 hydrochloride

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