Potent and selective adenosine A2B
receptor inverse agonist (Ki
values are 1.39, 157, 112 and 230 nM for human A2B
Soluble to 5 mM in DMSO
Store at +4°C
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Manufactured and sold under license from Adenosine Therapeutics, LLC
Anilide derivatives of an 8-phenylxanthine carboxylic congener are highly potent and selective antagonists at human A2B adenosine receptors.
Kim et al.
ZM241385, DPCPX, MRS1706 are inverse agonists with different relative intrinsic efficacies on constitutively active mutants of the human adenosine A2B receptor.
Li et al.
New developments in A1 and A2 adenosine receptor antagonists.
Kiec-Kononowicz et al.
Pure Appl.Chem., 2001;73:1411
The citations listed below are publications that use Tocris products. Selected citations for MRS 1706 include:
Showing Results 1 - 10 of 11