Nalmefene hydrochloride

Tocris Bioscience | Catalog # 4085

Opioid receptor antagonist
Tocris Bioscience

Key Product Details

Description

Opioid receptor antagonist
View all Miscellaneous/Non-selective Opioid Antagonists »

Product Description

Nalmefene hydrochloride is an opioid receptor antagonist; displays a longer half life than Naloxone. Exhibits neuroprotective effects after traumatic brain injury in the rat.

Product Specifications for Nalmefene hydrochloride

Molecular Weight

375.89

Formula

C21H25NO3.HCl

Storage

Desiccate at RT

Purity

≥98% (HPLC)

Chemical Name

(5α)-17-(Cyclopropylmethyl)-4,5-epoxy-6-methylenemorphinan-3,14-diol hydrochloride

CAS Number

58895-64-0

PubChem ID

5388881

InChI Key

GYWMRGWFQPSQLK-OPHZJPRHSA-N

SMILES

C=C3[C@H]5[C@]24C1=C(O5)C(O)=CC=C1C[C@@H](N(CC6CC6)CC4)[C@@](O)2CC3.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 37.59 100
DMSO 37.59 100

Preparing Stock Solutions for Nalmefene hydrochloride

The following data is based on the product molecular weight 375.89.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.66 mL 13.30 mL 26.60 mL
5 mM 0.53 mL 2.66 mL 5.32 mL
10 mM 0.27 mL 1.33 mL 2.66 mL
50 mM 0.05 mL 0.27 mL 0.53 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 9 publications citing the usage of this product.

Product Documents for Nalmefene hydrochloride

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Nalmefene hydrochloride

For research use only

Citations for Nalmefene hydrochloride

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