NVS MLLT-1

Catalog # Availability Size / Price Qty
7482/10
7482/50
NVS MLLT-1 | CAS No. 2561471-13-2 | Bromodomain Inhibitors
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Description: Selective MLLT1/3 inhibitor

Chemical Name: N-[2-[[(2S)-2-Methyl-1-pyrrolidinyl]methyl]-1H-benzimidazol-6-yl]-6-isoquinolinecarboxamide

Purity: ≥98%

Product Details
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Biological Activity

NVS-MLLT-1 is a selective inhibitor of YEATS domain of MLLT1 and MLLT3 (IC50 values are 150 and 254 nM for MLLT1 and MLLT3, respectively). It shows selectivity for YEATS2/4 domains and over all bromodomains (CERC2 IC50 > 40 μM).

Technical Data

M.Wt:
385.47
Formula:
C23H23N5O
Solubility:
Soluble to 100 mM in DMSO and to 50 mM in ethanol
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
2561471-13-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the NVS MLLT-1 probe summary on the SGC website.

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