Potent endogenous vanilloid TRPV1 (VR1) receptor agonist (EC50
= 36 nM at hVR1) with low affinity for rCB1
= 1.6 μ
M). Potently induces VR1-mediated thermal hyperalgesia in rats in vivo
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Anitallodynic effects of loperamide and fentanyl against topical capsaicin-induced allodynia in unanesthetized primates.
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