Chemical Name: (9Z)-N-[1-((R)-4-Hydroxbenzyl)-2-hydroxyethyl]-9-octadecenamide
Biological ActivityOMDM-2 is a metabolically stable inhibitor of anandamide cellular uptake (Ki = 3 μM). Displays relatively low affinity for CB1 and CB2 receptors (Ki values are 5.1 and > 10 μM) and for vanilloid VR1 receptors (EC50 = 10 μM). FABP inhibitor. Has minimal activity against FAAH (Ki > 50 μM). Active in vivo.
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Novel selective and metabolically stable inhibitors of anandamide cellular uptake.
Ortar et al.
In vivo pharmacological actions of two novel inhibitors of anandamide cellular uptake.
de Lago et al.
A personal retrospective: Elevating Anandamide (AEA) by targeting fatty acid amide hydrolase (FAAH) and the fatty acid binding proteins (FABPs).
Citation for OMDM-2
The citations listed below are publications that use Tocris products. Selected citations for OMDM-2 include:
1 Citation: Showing 1 - 1
Endocannabinoids acting at cannabinoid-1 receptors regulate cardiovascular function in hypertension.
Authors: Bátkai Et al.
FASEB J 2004;110:1996
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