PSNCBAM-1

Catalog # Availability Size / Price Qty
5321/50
5321/10
PSNCBAM-1 | CAS No. 877202-74-9 | Cannabinoid R1/CB1 Modulators
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Description: Negative allosteric modulator of CB1 receptors

Chemical Name: N-(4-Chlorophenyl)-N'-[3-[6-(1-pyrrolidinyl)-2-pyridinyl]phenyl]urea

Purity: ≥99%

Product Details
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Reviews (1)

Biological Activity

CB1 receptor negative allosteric modulator (IC50 values are 45 and 209 nM for the inhibition of CP 55,940 and WIN 55,212-2 respectively). Has no effect at the CB2 receptor. Decreases food intake and body weight in rats.

Technical Data

M.Wt:
392.88
Formula:
C22H21ClN4O
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
877202-74-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Works as described, another very interesting compound.
By Jonathan Fay on 05/30/2019
Application: Species: Human

Allosteric enhancement of radiolabeled agonist binding.

PMID: 24206272

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