RN 1 dihydrochloride

   
Product Datasheet
Catalog Number:4977
Chemical Name:1-(4-methyl-1-piperazinyl)-2-[[(1R*,2S*)-2-[4-phenylmethoxy)phenyl]cyclopropyl]amino]ethanone dihydrochloride
Product Details
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Biological Activity
Potent lysine specific demethylase 1 (LSD1) inhibitor (IC50 = 70 nM). Exhibits selectivity for LSD1 over MAO-A and MAO-B (IC50 values are 0.51 and 2.79 μM for MAO-A and MAO-B, respectively). Impairs long-term, but not short-term memory in mice. Brain penetrant following systemic administration.
Technical Data
  • M.Wt:
    452.42
  • Formula:
    C23H29N3O2.2HCl
  • Solubility:
    Soluble to 20 mM in water and to 20 mM in DMSO with gentle warming
  • Purity:
    >97
  • Storage:
    Store at -20°C
  • CAS No:
    1781835-13-9
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
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