SB 452533

  ( 1 citations )    
Product Datasheet
Catalog Number:3265
Chemical Name:N-(2-Bromophenyl)-N'-[2-[ethyl(3-methylphenyl)amino]ethyl]-urea
Product Details
Citations (1)
Supplemental Products
Reviews
Biological Activity
Potent TRPV1 antagonist against capsaicin (pKb = 7.7), noxious heat and acid-mediated (pIC50 = 7.0) receptor activation (pKi = 6.22 at the recombinant hTRPV1 receptor). Exhibits analgesic properties.
Technical Data
  • M.Wt:
    376.29
  • Formula:
    C18H22BrN3O
  • Solubility:
    Soluble to 100 mM in DMSO and to 10 mM in ethanol with gentle warming
  • Purity:
    >98
  • Storage:
    Store at RT
  • CAS No:
    459429-39-1
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Additional Information
Licensing Caveats:
Sold for research purposes only under agreement from GlaxoSmithKline
Product Datasheets
Citations:

The citations listed below are publications that use Tocris products. Selected citations for SB 452533 include:

1 Citations: Showing 1 - 1

  1. Measurement of Ensemble TRPV1 Ion Channel Currents Using Droplet Bilayers.
    Authors: Vijayvergiya Et al.
    Mol Pain  2015;10:e0141366

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Note: No more than 500 mg per individual per year to be sold without prior permission from the licence holder.
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