SER 601

Key Product Details

Product Description

Potent and selective CB₂ receptor agonist (K_i values are 6.3 nM and 1.2 μM for CB₂ and CB₁ receptors respectively). Displays analgesic activity in the formalin test in mice.

Product Specifications for SER 601

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Preparing Stock Solutions for SER 601

The following data is based on the product molecular weight 434.61.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

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Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.5 mM	4.60 mL	23.01 mL	46.02 mL
2.5 mM	0.92 mL	4.60 mL	9.20 mL
5 mM	0.46 mL	2.30 mL	4.60 mL
25 mM	0.09 mL	0.46 mL	0.92 mL

Calculators

Background References

References are publications that support the biological activity of the product. See our Citations tab to view 3 publications citing the usage of this product.

• Contartese A novel CB2 agonist, COR167, potently protects rat brain cortical slices against OGD and reperfusion injury. Pharmacol.Res. 2012 PMID: 23036353
• Pasquini Investigations on the 4-quinolone-3-carboxylic acid motif. 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo. J.Med.Chem. 2008 PMID: 18680276

Product Documents for SER 601