SGC GAK 1
Chemical Name: 6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine
Biological ActivityHigh affinity cyclin G associated kinase (GAK) inhibitor (Kd = 1.9 nM). Exhibits >30-fold selectivity for GAK over a panel of other kinases. Inhibits GAK in live cell assays (IC50 = 110 nM).
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
SGC-GAK-1: a chemical probe for cyclin G associated kinase (GAK).
Asquith et al.
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