SGC GAK 1

   
Product Datasheet
Catalog Number:6564
Chemical Name:6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine
Product Details
Reviews
Biological Activity
High affinity cyclin G associated kinase (GAK) inhibitor (Kd = 1.9 nM). Exhibits >30-fold selectivity for GAK over a panel of other kinases. Inhibits GAK in live cell assays (IC50 = 110 nM).
Technical Data
  • M.Wt:
    389.24
  • Formula:
    C18H17BrN2O3
  • Solubility:
    Soluble to 100 mM in DMSO and to 50 mM in ethanol
  • Purity:
    >99
  • Storage:
    Store at -20°C
  • CAS No:
    2226517-76-4
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Additional Information
Licensing Caveats:
This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the SGC GAK 1 probe summary on the SGC website.
Product Datasheets

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