SGC GAK 1

Catalog # Availability Size / Price Qty
6564/5
6564/25
Cat.No. 6564 - SGC GAK 1 | C18H17BrN2O3 | CAS No. 2226517-76-4
1 Image
Description: High affinity cyclin G associated kinase (GAK) inhibitor

Chemical Name: 6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine

Purity: ≥99%

Product Details
Reviews

Biological Activity

High affinity cyclin G associated kinase (GAK) inhibitor (Kd = 1.9 nM). Exhibits >30-fold selectivity for GAK over a panel of other kinases. Inhibits GAK in live cell assays (IC50 = 110 nM).

Technical Data

M.Wt:
389.24
Formula:
C18H17BrN2O3
Solubility:
Soluble to 100 mM in DMSO and to 50 mM in ethanol
Purity:
≥99%
Storage:
Store at -20°C
CAS No:
2226517-76-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.

Additional Information

Licensing Caveats:
This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the SGC GAK 1 probe summary on the SGC website.

Product Datasheets

Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Molarity Calculator

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / CoA (available online).

FAQs

No product specific FAQs exist for this product, however you may

View all Small Molecule FAQs

Reviews for SGC GAK 1

There are currently no reviews for this product. Be the first to review SGC GAK 1 and earn rewards!

Have you used SGC GAK 1?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥1250 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.