Protease-activated receptor 2 (PAR2
) agonist (Ki
= 9.64 μ
M and IC50
= 10.4 μ
M). Corresponds to the tethered ligand exposed by trypsin cleavage of PAR-2. Control peptide VKGILS-NH2
also available (Cat. No. 3392).
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Other Product-Specific Information:
Molecular cloning, expression and potential functions of the human proteinase-activated receptor-2.
Bohm et al.
International union of pharmacology XXVIII. Proteinase-activated receptors.
Hollenberg and Compton
Binding of a highly potent protease-activated receptor-2 (PAR2) activating peptide, [3H]2-furoyl-LIGRL-NH2, to human PAR2.
Kanke et al.
The citations listed below are publications that use Tocris products. Selected citations for SLIGKV-NH2 include:
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