Potent FAAH inhibitor; (IC50
values are 0.28 and 0.72 nM, at rat and human FAAH respectively). Displays analgesic effects in vivo
models of neuropathic and inflammatory pain. Brain penetrant.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Design, synthesis, and biological evaluation of a series of piperazine ureas as fatty acid amide hydrolase inhibitors.
Kono et al.