Discontinued Product

5139 has been discontinued.
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Telmisartan | CAS No. 144701-48-4 | Angiotensin AT1 Receptor Antagonists
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Description: AT1 antagonist; PPARγ partial agonist

Chemical Name: 4'-[(1,4'-Dimethyl-2'-propyl[2,6'-bi-1H-benzimidazol]-1'-yl)methyl]-[1,1'-biphenyl]-2-carboxylic acid

Purity: ≥99%

Product Details
Citations (1)

Biological Activity

Telmisartan is an antagonist of the angiotensin II type 1 receptor (AT1) (Ki = 3.7 nM). Exhibits antihypertensive activity in a renin-dependent model of hypertension. Partial agonist of PPARγ receptors; shown to improve insulin sensitivity in rodents receiving high fat diets.

Technical Data

Soluble to 20 mM in DMSO
Store at RT

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citation for Telmisartan

The citations listed below are publications that use Tocris products. Selected citations for Telmisartan include:

1 Citation: Showing 1 - 1

  1. Development of telmis. in the therapy of spinal cord injury: pre-clinical study in rats.
    Authors: Lin Et al.
    Psychopharmacology (Berl)  2015;9:4709


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