TP 003

Catalog # Availability Size / Price Qty
4414/10
4414/50
Cat.No. 4414 - TP 003 | C23H16F3N3O | CAS No. 628690-75-5
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Description: Functionally selective GABAA (α3 subtype) partial agonist

Chemical Name: 2',4-Difluoro-5'-[8-fluoro-7-(1-hydroxy-1-methylethyl)imidazo[1,2-a]-pyridin-3-yl]-[1,1'-biphenyl]-2-carbonitrile

Purity: ≥98%

Product Details
Citations (1)
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Biological Activity

Functionally selective GABAA receptor (α3 subtype) partial agonist. Exhibits affinity for the benzodiazepine binding site on human GABAA receptors. Potentiates the GABA (α3 subtype) response selectively with high efficacy. Produces anxiolytic-like effects in rodent behavioral models of anxiety.

Technical Data

M.Wt:
407.39
Formula:
C23H16F3N3O
Solubility:
Soluble to 100 mM in DMSO and to 50 mM in ethanol
Purity:
≥98%
Storage:
Store at +4°C
CAS No:
628690-75-5

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.

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Citation for TP 003

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