UCM 707

Name: UCM 707
Brand: Tocris Bioscience
SKU: 1966

Catalog #: 1966 Datasheet / COA / SDS

Discontinued Product

1966 has been discontinued.

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UCM 707 | CAS No. 390824-20-1 | Cannabinoid Transporter Inhibitors

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Description: Potent anandamide transport inhibitor

Chemical Name: (5Z,8Z,11Z,14Z)-N-(3-Furanylmethyl)-5,8,11,14-eicosatetraenamide

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Product Details

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Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

UCM 707 is a potent endocannabinoid transport inhibitor. IC₅₀ values are 0.8 and 30 μM for inhibition of the anandamide transporter and FAAH respectively. K_i values are 4700, 67 and > 5000 nM for CB₁, CB₂and VR1 receptors respectively. Potentiates hypokinetic and antinociceptive effects of anandamide in vivo.

Technical Data

M.Wt:

383.57

Formula:

C₂₅H₃₇NO₂

Solubility:

Soluble to 100 mM in ethanol and to 100 mM in DMSO

Storage:

Desiccate at -20°C

CAS No:

390824-20-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

Design, synthesis and biological evaluation of new endocannabinoid transporter inhibitors.
Lopez-Rodriguez et al.
Eur.J.Med.Chem., 2003;38:403
Design, synthesis, and biological evaluation of new inhibitors of the endocannabinoid uptake: comparison with effects on fatty acid amidohydrolase.
Lopez-Rodriguez et al.
J.Med.Chem., 2003;46:1512

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