YM 022

Catalog # Availability Size / Price Qty
1408/10
1408/50

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YM 022 | CAS No. 145084-28-2 | CCK2 Receptor Antagonists
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Description: Highly potent, selective non-peptide CCK2 antagonist

Chemical Name: (R)-N-[2,3-Dihydro-1-[2-(2-methylphenyl)-2-oxoethyl]-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl]-N'-(3-methylphenyl)-urea

Purity: ≥99%

Product Details
Citations (4)
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Biological Activity

YM 022 is an extremely potent and highly selective non-peptide CCK2 silent antagonist (Ki values are 68 pM and 63 nM at CCK2 and CCK1 receptors respectively). Acts in vivo to potently inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation with a long duration of action.

Technical Data

M.Wt:
516.6
Formula:
C32H28N4O3
Solubility:
Soluble to 100 mM in DMSO and to 10 mM in ethanol
Purity:
≥99%
Storage:
Store at RT
CAS No:
145084-28-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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