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2 results for "GPR55 Receptor Antagonists Small Molecules and Peptides" in Products
GPR55 Receptor Antagonists Small Molecules and Peptides
GPR55 is a previously orphan receptor that exhibits affinity for endogenous, plant and synthetic cannabinoids, as well as lysophosphatidylinositols (LPIs), which are suggested to be its endogenous ligand. The effects of cannabinoid ligands that are inactive at CB1 and CB2, e.g. palmitoylethanolamide, are thought to be mediated through GPR55.
GPR55 is coupled to both the Gα12/13 and the Gαq intracellular pathways and displays complex pharmacology, with ligands having functional ...
Potent, selective GPR55 antagonist
| Alternate Names: | CID 1261822 |
| Chemical Name: | N-[4-[[(3,4-Dimethyl-5-isoxazolyl)amino]sulfonyl]phenyl]-6,8-dimethyl-2-(2-pyridinyl)-4-quinolinecarboxamide |
| Purity: | ≥98% |
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Selective GPR55 antagonist
| Chemical Name: | 4-[4,6-Dihydro-4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxopyrrolo[3,4-c]pyrazol-5(1H)-yl]benzoic acid |
| Purity: | ≥98% |
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