3 results for "MAPKAPK2 Small Molecules and Peptides" in Products

MAPKAPK2 Small Molecules and Peptides

Potent MK2 inhibitor

Chemical Name: (10R)-9,10,11,12-Tetrahydro-10-methyl-3-(6-methyl-3-pyridinyl)-8H-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one
Purity: ≥98%
Potent MK2 inhibitor
Loading...

Cdk inhibitor; potently inhibits cdk9; also inhibits MK2

Chemical Name: 1,5,6,7-Tetrahydro-2-(4-pyridinyl)-4H-pyrrolo[3,2-c]pyridin-4-one hydrochloride
Purity: ≥98%
Cdk inhibitor; potently inhibits cdk9; also inhibits MK2
Loading...

Potent and selective p38α and p38β Degrader (PROTAC®); active in vivo

Chemical Name: 3-(3-Bromo-4-((2,4-difluorobenzyl)oxy)-6-methyl-2-oxopyridin-1(2H)-yl)-N-(4-(1-(4-((4-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)butyl)amino)-4-oxobutyl)-1H-1,2,3-triazol-4-yl)butyl)-4-methylbenzamide
Purity: ≥97%
Potent and selective p38α and p38β Degrader (PROTAC®); active in vivo
Loading...
Results Per Page
5 10 25 50
  • / 1