5 results for "Cannabinoid R1/CB1 Antagonists Small Molecules and Peptides" in 产品
Cannabinoid R1/CB1 Antagonists Small Molecules and Peptides
The CB1 receptor, also known as the central cannabinoid receptor, is a member of the cannabinoid receptor group of G-protein-coupled receptors that also includes CB2 and GPR55. CB1 receptors are found mainly in the terminals of central and peripheral neurons, where they usually mediate inhibition of neurotransmitter release. They can also be present on some non-neuronal cells, including immune cells.
CB1 receptor antagonists are drugs that bind to the CB1 receptor and prevent its activation ...
Potent CB1 antagonist; also GPR55 agonist
| Chemical Name: | N-(Piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide |
| Purity: | ≥98% |
CB1 antagonist
| Chemical Name: | 1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-4-(ethylamino)piperidine-4-carboxamide hydrochloride |
| Purity: | ≥98% |
High affinity and selective CB1 antagonist
| Chemical Name: | 5-[4-(4-Cyano-1-butyn-1-yl)phenyl]-1-(2,4-dichlorophenyl)-N-(1,1-dioxido-4-thiomorpholinyl)-4-methyl-1H-pyrazole-3-carboxamide |
| Purity: | ≥98% |
Ultra-high affinity and selective CB1 antagonist
| Chemical Name: | 8-Chloro-1-(2,4-dichlorophenyl)-1,4,5,6-tetrahydro-N-1-piperidinyl-benzo[6,7]cyclohepta[1,2-c]pyrazole-3-carboxamide |
| Purity: | ≥98% |
High affinity and selective CB1 antagonist
| Chemical Name: | 5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide |
| Purity: | ≥98% |
