4 results for "Glucocorticoid Receptor Agonists" in 产品

Glucocorticoid Receptor Agonists

Glucocorticoid Receptor (GR), also known as NR3C1, is a member of the NR3 family of nuclear receptors. It mediates the physiological and pharmacological actions of glucocorticoids. GR is a modular protein that is composed of three major domains: a N-terminal transactivation domain (NTD, amino acids [aa] 1-421); a central DNA-binding domain (DBD, aa...

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Selective high affinity glucocorticoid receptor agonist

Chemical Name: (6α,11β,16α,17α)-6,9-Difluoro-11-hydroxy-16-methyl-3-oxo-17-(1-oxopropoxy)androsta-1,4-diene-17-carbothioic acid fluoromethyl ester
Purity: ≥98%
Selective high affinity glucocorticoid receptor agonist
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Glucocorticoid receptor agonist

Chemical Name: N-[4-[1-(4-Fluorophenyl)-1H-indazol-5-yl-3-(trifluoromethyl)phenyl]benzenesulfonamide
Purity: ≥98%
Glucocorticoid receptor agonist
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Glucocorticoid receptor agonist

Chemical Name: 11β,17β,21-Trihydroxy-6α-methyl-1,4-pregnadiene-3,20-dione
Purity: ≥98%
Glucocorticoid receptor agonist
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Endogenous glucocorticoid

Chemical Name: (11β)-11,21-Dihydroxypregn-4-ene-3,20-dione
Purity: ≥98%
Endogenous glucocorticoid
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