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Kir6 blocker; non-hydrolyzable AMP analog
Kir6 (KATP) channel blocker
H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker
Kir 7.1 inhibitor; also inhibits Kir 6.2
Selective blocker of inward-rectifier K+ channels
Vascular Kir6 (KATP) channel blocker
Kir6 (KATP) channel blocker
Kir6 (KATP) blocker; displays high affinity for SUR1/Kir6.2 channels