244 results for "P2X7/P2RX7" in 产品

P2X7/P2RX7 Products

P2RX7 belongs to the family of purinoceptors for ATP. It functions as a ligand-gated ion channel and is responsible for ATP-dependent lysis of macrophages through the formation of membrane pores permeable to large molecules. P2RX7 antagonists have emerged as novel therapeutics for the treatment of acute inflammation, pain and fever, with wider anti-inflammatory activity than currently used cyclooxygenase inhibitors.

Photoaffinity label for ATPase; also P2X7 agonist and P2X1/P2Y1 partial agonist

Chemical Name: 2'(3')-O-(4-Benzoylbenzoyl)adenosine-5'-triphosphate tri(triethylammonium) salt
Purity: ≥95%
Photoaffinity label for ATPase; also P2X7 agonist and P2X1/P2Y1 partial agonist
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Competitive P2X7 antagonist

Chemical Name: 3-[[5-(2,3-Dichlorophenyl)-1H-tetrazol-1-yl]methyl]pyridine hydrochloride
Purity: ≥98%
Competitive P2X7 antagonist
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Potent and selective P2X7 antagonist

Chemical Name: N-[1-[[(Cyanoamino)(5-quinolinylamino)methylene]amino]-2,2-dimethylpropyl]-3,4-dimethoxybenzeneacetamide
Purity: ≥97%
Potent and selective P2X7 antagonist
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Reactivity: Human, Mouse, Rat, Monkey
Details: Rabbit IgG Polyclonal
Applications: IHC, WB
Western Blot: P2X7/P2RX7 Antibody [NBP1-20180]
(15)
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Reactivity: Human, Mouse
Details: Goat IgG Polyclonal
Applications: IHC, WB, ELISA, ICC/IF
Western Blot: P2X7/P2RX7 Antibody [NBP1-37775]
(3)
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Non-competitive P2X7 antagonist

Chemical Name: 4-[(2S)-2-[(5-isoquinolinylsulfonyl)methylamino]-3-oxo-3-(4-phenyl-1-piperazinyl)propyl] phenyl isoquinolinesulfonic acid ester
Purity: ≥98%
Non-competitive P2X7 antagonist
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Reactivity: Human
Details: Mouse IgG2B Monoclonal Clone #7G1D6
Applications: IHC, WB, ELISA, Flow
Western Blot: P2X7/P2RX7 Antibody (7G1D6)BSA Free [NBP2-61748]
(6)
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Reactivity: Human, Mouse, Rat
Details: Rabbit IgG Polyclonal
Applications: IHC
Immunohistochemistry-Paraffin: P2X7/P2RX7 Antibody [NBP1-32470]
(3)
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Potent and selective human P2X7 antagonist

Chemical Name: 3-[1-[[(3'-Nitro[1,1'-biphenyl]-4-yl)oxy]methyl]-3-(4-pyridinyl)propyl]-2,4-thiazolidinedione
Purity: ≥98%
Potent and selective human P2X7 antagonist
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Potent P2X7 antagonist

Chemical Name: N-[2-[[2-[(2-Hydroxyethyl)amino]ethyl]amino]-5-quinolinyl]-2-tricyclo[3.3.1.13,7]dec-1-ylacetamide dihydrochloride
Purity: ≥98%
Potent P2X7 antagonist
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Reactivity: Human
Details: Mouse IgG2A Monoclonal Clone #CL11508
Applications: IHC, WB
Western Blot: P2X7/P2RX7 Antibody [NBP3-21196] -
(5)
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Potent and selective P2X7 antagonist

Chemical Name: N-Cyano-N"-[(1S)-1-phenylethyl]-N'-5-quinolinyl-guanidine
Purity: ≥98%
Potent and selective P2X7 antagonist
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Reactivity: Human, Mouse, Rat
Details: Rabbit IgG Polyclonal
Applications: IHC
Immunohistochemistry-Paraffin: P2X7/P2RX7 Antibody [NBP2-19654]
(4)
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Reactivity: Human
Details: Mouse IgG2A Monoclonal Clone #CL11508
Applications: IHC, WB
P2X7/P2RX7 Antibody (CL11508) - Azide and BSA Free Immunohistochemistry-Paraffin: P2X7/P2RX7 Antibody [NBP3-44150]
(5)
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Cell-permeable protein kinase C inhibitor

Chemical Name: 1,2-Dimethoxy-12-methyl[1,3]benzodioxolo[5,6-c]phenanthridinium chloride
Purity: ≥98%
Cell-permeable protein kinase C inhibitor
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Potent and selective P2X7 antagonist; brain penetrant

Chemical Name: 2-(Phenylthio)-N-[[tetrahydro-4-(4-phenyl-1-piperazinyl)-2H-pyran-4-yl]methyl-3-pyridinecarboxamide
Purity: ≥98%
Potent and selective P2X7 antagonist; brain penetrant
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Reactivity: Human
Details: Mouse IgG2A Monoclonal Clone #1058613
Applications: Flow
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Reactivity: Human
Details: Rabbit IgG Polyclonal
Applications: IHC, WB
Western Blot: P2X7/P2RX7 Antibody [NBP1-82738]
(3)
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Reactivity: Human
R&D Systems VersaClone cDNA Plasmids
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Reactivity: Rat
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Reactivity: Human
Source: Wheat germ
Applications: WB, ELISA, AP, DB, MA
SDS-PAGE: Recombinant Human P2X7/P2RX7 GST (N-Term) Protein [H00005027-P01]
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