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TRPV antagonist; also activator of ENaCδ
Potent and selective TRPV1 competitive antagonist
Potent and selective TRPV4 antagonist; orally active
Non-selective CaV2.1 and 2.2 blocker; also blocks TRPV channels
Potent and selective TRPV4 antagonist
Selective TRPV3 antagonist; brain penetrant
Antiallergic; inhibits inflammatory mediator release from mast cells
Potent and selective TRPV1 competitive antagonist
Reversible, competitive and potent TRPV1 antagonist
Potent and selective TRPV1 antagonist
Potent and selective TRPV1 antagonist
Potent and selective TRPV4 antagonist
Selective TRPV4 antagonist
Selective TRPV2 antagonist
