endothelin receptor antagonist (Ki
values are 1.4 and 1500 nM at ETA
receptors respectively). Reduces ischemia-induced ventricular arrhythmias in a rat model.
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Role of endothelin in cardiovascular disease.
Agapitov and Haynes
J.Renin Angiotensin Aldosterone Syst., 2002;3:1
Effects of selective ETB-receptor stimulation on arterial, venous and capillary functions in cat skeletal muscle.
Ekelund et al.
Distinct subdomains of human endothelin receptors determine their selectivity to endothelinA-selective antagonist and endothelinB-selective agonists.
Sakamoto et al.
Effect of a novel bifunctional endothelin receptor antagonist, IRL 3630A, on guinea pig respiratory mechanics.
Makatani et al.
The citations listed below are publications that use Tocris products. Selected citations for BQ-123 include:
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