Selective vanilloid receptor antagonist (Ki
= 3.2 μ
M). Inhibits carrageenan inflammation-induced hyperalgesic responses in the rat. Also activates amiloride-sensitive epithelial Na+
. Also available as part of the Vanilloid TRPV1 Receptor Tocriset™
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Selective antagonism of capsaicin by capsazepine: evidence for a spinal receptor site in capsaicin-induced antinociception.
Dickenson and Dray
A capsaicin-receptor antagonist, capsazepine, reduces inflammation-induced hyperalgesic responses in the rat: evidence for an endogenous capsaicin-like substance.
Kwak et al.
Capsazepine is a novel activator of the δ subunit of the human epithelial Na+ channel.
Yamamura et al.
The citations listed below are publications that use Tocris products. Selected citations for Capsazepine include:
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