Galeterone

Catalog # Availability Size / Price Qty
6108/10
6108/50
Cat.No. 6108 - Galeterone | C26H32N2O | CAS No. 851983-85-2
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Description: CYP17 inhibitor; also androgen receptor antagonist
Alternative Names: TOK-001, VN/124-1

Chemical Name: (3β)-17-(1H-Benzimidazol-1-yl)androsta-5,16-dien-3-ol

Purity: ≥98%

Product Details
Reviews

Biological Activity

CYP17 inhibitor (IC50 = 300 nM) and androgen receptor antagonist (IC50 = 384 nM in PC3-AR cells). Inhibits DHT-stimulated prostate cancer cell proliferation in vitro. Exhibits antitumor activity in SCID mice bearing prostate cancer xenografts.

Technical Data

M.Wt:
388.55
Formula:
C26H32N2O
Solubility:
Soluble to 50 mM in DMSO and to 50 mM in ethanol
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
851983-85-2

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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