Cytochrome P450 Inhibitors: Products

Blocks retinoic acid metabolism

11-β hydroxylase inhibitor

Cytochrome P450c17 inhibitor

Potent aromatase (CYP19) inhibitor

Steroidal aromatase (CYP19) inhibitor

Cytochrome P450 inhibitor; antifungal

Potent, reversible non-steroidal aromatase inhibitor

CYP17 inhibitor; also androgen receptor antagonist

Allosteric Calcium-sensing receptor (CaSR) agonist; also CYP2D2 inhibitor and Ca2+ channel blocker; orally bioavailable

Potent CYP17A1 inhibitor