A selective competitive 5-HT1B
) silent antagonist with pKB
values of 7.3 and 6.3 for human cloned 5-HT1B
receptors respectively and only weak binding at a number of other 5-HT subtypes.
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Evidence for 5-HT1-like receptor-mediated vasoconstriction in human pulmonary artery.
MacLean et al.
The activity of 5-HT1D receptor ligands at cloned human 5-HT1Dα and 5-HT1Dβ receptors.
Walsh et al.
Use of GR55562, a selective 5-HT1D antagonist, to investigate 5-HT1D receptor subtypes mediating cerebral vasoconstriction.
Connor et al.
The citations listed below are publications that use Tocris products. Selected citations for GR 55562 dihydrochloride include:
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