JNJ 17203212

Catalog # Availability Size / Price Qty
3361/10
3361/50
TRPV Antagonists Small Molecule
1 Image
Description: Reversible, competitive and potent TRPV1 antagonist

Chemical Name: 4-[3-(Trifluoromethyl)-2-pyridinyl]-N-[5-(trifluoromethyl)-2-pyridinyl]-1-piperazinecarboxamide

Purity: ≥99%

Product Details
Citations (2)
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Biological Activity

Reversible, competitive and potent TRPV1 antagonist (pKi values are 6.5, 7.1 and 7.3 at rat, guinea pig and human TRPV1 respectively). Inhibits capsaicin- and H+-induced channel activation (pIC50 values are 6.32 and 7.23 respectively) and exhibits antitussive and analgesic activity in vivo.

Technical Data

M.Wt:
419.32
Formula:
C17H15F6N5O
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
821768-06-3

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for JNJ 17203212

The citations listed below are publications that use Tocris products. Selected citations for JNJ 17203212 include:

2 Citations: Showing 1 - 2

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