KT 5823

Catalog # Availability Size / Price Qty
1289/100U
KT 5823 | CAS No. 126643-37-6 | Protein Kinase G Inhibitors
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Description: Selective protein kinase G inhibitor

Chemical Name: (9S,10R,12R)-2,3,9,10,11,12-Hexahydro-10-methoxy-2,9-dimethyl-1-oxo-9,12-epoxy-1H-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-10-carboxylic acid, methyl ester

Purity: ≥98%

Product Details
Citations (5)
Reviews

Biological Activity

Selective inhibitor of protein kinase G (Ki values are 0.23, 4 and > 10 μM for inhibition of PKG, PKC and PKA respectively). Inhibits SNP-stimulated PKG activity with an IC50 of 60 nM in dispersed smooth muscle cells and has little effect on PKA activity at concentrations of up to 10 μM.

Technical Data

M.Wt:
495.53
Formula:
C29H25N3O5
Solubility:
Soluble to 50 mM in DMSO
Purity:
≥98%
Storage:
Desiccate at -20°C
CAS No:
126643-37-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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