NNC 26-9100

Tocris Bioscience | Catalog # 2440

Selective sst4 agonist
Tocris Bioscience
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Key Product Details

Description

Selective sst4 agonist

Product Description

NNC 26-9100 is a somatostatin sst4 receptor agonist that displays > 100-fold selectivity over sst2 receptors (Ki values are 6 and 621 nM for sst4 and sst2 receptors respectively). Potently inhibits forskolin-induced cAMP accumulation (EC50 = 26 nM).

Product Specifications for NNC 26-9100

Molecular Weight

556.35

Formula

C22H25N6Cl2SBr

Storage

Store at +4°C

Purity

≥98% (HPLC)

Chemical Name

1-[3-[N-(5-Bromopyridin-2-yl)-N-(3,4-dichlorobenzyl)amino]propyl]-3-[3-(1H-imidazol-4-yl)propyl]thiourea

CAS Number

199522-35-5

PubChem ID

9893924

InChI Key

UREJDUPKGMFJRU-UHFFFAOYSA-N

SMILES

ClC1=C(Cl)C=C(CN(CCCNC(=S)NCCCC2=CNC=N2)C2=CC=C(Br)C=N2)C=C1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

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Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
DMSO 27.82 50
Ethanol 27.82 50

Preparing Stock Solutions for NNC 26-9100

The following data is based on the product molecular weight 556.35.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.5 mM 3.59 mL 17.97 mL 35.95 mL
2.5 mM 0.72 mL 3.59 mL 7.19 mL
5 mM 0.36 mL 1.80 mL 3.59 mL
25 mM 0.07 mL 0.36 mL 0.72 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 3 publications citing the usage of this product.

Product Documents for NNC 26-9100

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for NNC 26-9100

For research use only

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