PF 4800567 hydrochloride

Catalog # Availability Size / Price Qty
4281/10
4281/50
Casein Kinase 1 Inhibitors Small Molecule
1 Image
Description: Selective casein kinase 1ε inhibitor

Chemical Name: 3-[(3-Chlorophenoxy)methyl]-1-(tetrahydro-2H-pyran-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine hydrochloride

Purity: ≥99%

Product Details
Citations (4)
Reviews

Biological Activity

Selective casein kinase 1ε inhibitor; displays 22-fold greater potency towards CK1ε than CK1δ (IC50 values are 32 and 711 nM for CK1ε and CK1δ respectively). ATP competitive. Displays minimal effect on the circadian clock.

External Portal Information

Chemicalprobes.org is a portal that offers independent guidance on the selection and/or application of small molecules for research. The use of PF 4800567 is reviewed on the chemical probes website.

Technical Data

M.Wt:
396.27
Formula:
C17H18ClN5O2.HCl
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥99%
Storage:
Desiccate at RT
CAS No:
1391052-28-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold for research purposes under agreement from Pfizer Inc.

Product Datasheets

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Citations for PF 4800567 hydrochloride

The citations listed below are publications that use Tocris products. Selected citations for PF 4800567 hydrochloride include:

4 Citations: Showing 1 - 4

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