R-96544 hydrochloride

Catalog # Availability Size / Price Qty
1742/10
1742/50
R-96544 hydrochloride | CAS No. 167144-80-1 | 5-HT2A Receptor Antagonists
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Description: Potent, selective 5-HT2A antagonist

Chemical Name: (2R,4R)-5-[2-[2-[2-(3-Methoxyphenyl)ethyl]phenoxy]ethyl]-1-methyl-3-pyrrolidinol hydrochloride

Product Details
Citations (3)
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Biological Activity

Potent, selective 5-HT2 receptor antagonist; displays some selectivity for 5-HT2A receptors (Ki = 1.6 nM). IC50 values are 2.2, 310, 2400, 3700, > 5000 and > 5000 nM for 5-HT2, α1-adrenergic, D2 dopamine, 5-HT1, 5-HT3 and β-adrenergic receptors respectively. Inhibits 5-HT-induced platelet aggregation and pressor responses in vivo.

Technical Data

Formula:
C22H29NO3.HCl
Solubility:
Soluble to 100 mM in water and to 100 mM in DMSO
Storage:
Store the unopened product at room temperature. Do not use past expiration date.
CAS No:
167144-80-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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Citations for R-96544 hydrochloride

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