Potent, selective 5-HT
receptor antagonist; displays some selectivity for 5-HT
= 1.6 nM). IC
values are 2.2, 310, 2400, 3700, > 5000 and > 5000 nM for 5-HT
-adrenergic receptors respectively. Inhibits 5-HT-induced platelet aggregation and pressor responses
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Pharmacological profiles of R-96544, the active form of a novel 5-HT 2A receptor antagonist R-102444.
Ogawa et al.
Effects of R-102444 and its active metabolite R-96544, selective 5-HT 2A receptor antagonists, on experimental acute and chronic pancreatitis: additional evidence for possible involvement of 5-HT 2A receptors in the development of expe
Ogawa et al.
[2-(ω-Phenylalkyl)phenoxy]alkylamines III: Synthesis and selective serotonin-2 receptor binding.
Tanaka et al.
The citations listed below are publications that use Tocris products. Selected citations for R-96544 hydrochloride include:
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