LSD1 inhibitor (IC50
= 990 nM; Ki
= 610 nM). Exhibits selectivity for LSD1 over MAO-B and MAO-A (Ki
values are 17 and 110 μ
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Structurally designed trans-2-phenylcyclopropylamine derivatives potently inhibit histone demethylase LSD1/KDM1.
Mimasu et al.