SB 222200

Catalog # Availability Size / Price Qty
1393/10
1393/50
SB 222200 | CAS No. 174635-69-9 | NK3 Receptor Antagonists
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Description: Potent, selective non-peptide NK3 antagonist. Brain penetrant

Chemical Name: 3-Methyl-2-phenyl-N-[(1S)-1-phenylpropyl]-4-quinolinecarboxamide

Purity: ≥98%

Product Details
Citations (2)
Supplemental Products
Reviews (1)

Biological Activity

SB 222200 is a potent and selective non-peptide NK3 receptor antagonist (Ki values are 4.4, > 100,000 and 250 nM for human NK3, NK1 and NK2 receptors respectively). Antihypertensive in vivo. Brain penetrant.

Technical Data

M.Wt:
380.48
Formula:
C26H24N2O
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Purity:
≥98%
Storage:
Store at RT
CAS No:
174635-69-9

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold under license

Product Datasheets

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Citations for SB 222200

The citations listed below are publications that use Tocris products. Selected citations for SB 222200 include:

2 Citations: Showing 1 - 2

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