TC-G 1004

Catalog # Availability Size / Price Qty
4407/10
4407/50
TC-G 1004 | CAS No. 1061747-72-5 | Adenosine A2a Receptor Antagonists
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Description: Potent and selective A2A antagonist

Chemical Name: N-[2-(3,5-Dimethyl-1H-pyrazol-1-yl)-6-[6-(4-methoxy-1-piperidinyl)-2-pyridinyl]-4-pyrimidinyl]acetamide

Purity: ≥98%

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Biological Activity

TC-G 1004 is a potent antagonist of adenosine A2A receptors; displays >100-fold selectivity for A2A over A1 receptors (Ki values are 0.44 and 85 nM respectively). Potentiates L-DOPA-induced rotational behavior in 6-OHDA-lesioned rats.

Technical Data

M.Wt:
421.5
Formula:
C22H27N7O2
Solubility:
Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
1061747-72-5

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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