TC-N 1752

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TC-N 1752 | CAS No. 1211866-85-1 | Voltage-gated Sodium Channel Blockers
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Description: NaV channel blocker

Chemical Name: N-[2-Methyl-3-[[4-[4-[[4-(trifluoromethoxy)phenyl]methoxy]-1-piperidinyl]-1,3,5-triazin-2-yl]amino]phenyl]acetamide

Purity: ≥99%

Product Details
Citations (1)
Reviews

Biological Activity

Human NaV channel inhibitor (IC50 values are 0.17, 0.3, 0.4, 1.1 and 1.6 μM at hNaV1.7, hNaV1.3, hNaV1.4, hNaV1.5 and hNav1.9 respectively). Also inhibits tetrodotoxin-sensitive sodium channels. Displays analgesic efficacy in the formalin pain model.

Technical Data

M.Wt:
516.52
Formula:
C25H27F3N6O3
Solubility:
Soluble to 100 mM in DMSO and to 10 mM in 1eq. HCl
Purity:
≥99%
Storage:
Store at +4°C
CAS No:
1211866-85-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

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Citation for TC-N 1752

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