Biological Activity Human NaV channel inhibitor (IC50 values are 0.17, 0.3, 0.4, 1.1 and 1.6 μM at hNaV1.7, hNaV1.3, hNaV1.4, hNaV1.5 and hNav1.9 respectively). Also inhibits tetrodotoxin-sensitive sodium channels. Displays analgesic efficacy in the formalin pain model.
Soluble to 100 mM in DMSO and to 10 mM in 1eq. HCl
Store at +4°C
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For batch specific data refer to the Certificate of Analysis.
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