Catalog Number: 4069
Chemical Name: (5R)-5-[(3S)-3-Hydroxy-4-phenyl-1-buten-1-yl]-1-[6-(2H-tetrazol-5-yl)hexyl]-2-pyrrolidinone
Biological Activity
Highly selective EP4 agonist (EC50 = 2.5 nM; Ki = 1.2 nM). Displays no significant binding at other prostaglandin receptors at concentrations up to 14 μM.
Technical Data
  • M.Wt:
    383.49
  • Formula:
    C21H29N5O2
  • Solubility:
    Soluble in ethanol (supplied pre-dissolved in anhydrous ethanol, 5mg/ml)
  • Purity:
    >98%
  • Storage:
    Store at -20°C
  • CAS No:
    346673-06-1
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.
Background References
  1. Discovery of a potent and selective agonist of the prostaglandin EP4 receptor.
    Billot et al.
    Bioorg.Med.Chem.Lett., 2003;130:1129
Citations:

The citations listed below are publications that use Tocris products. Selected citations for TCS 2510 include:

1 Citations: Showing 1 - 1

  1. Prostaglandin E(2) mediates proliferation and chloride secretion in ADPKD cystic renal epithelia.
    Authors: Liu Et al.
    Am J Physiol Renal Physiol 2012;303:F1425

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