VU 0255035

Catalog # Availability Size / Price Qty
3727/25
3727/5
Cat.No. 3727 - VU 0255035 | C18H20N6O3S2 | CAS No. 1135243-19-4
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Description: Highly selective M1 antagonist

Chemical Name: N-[3-Oxo-3-[4-(4-pyridinyl)-1-piperazinyl]propyl]-2,1,3-benzothiadiazole-4-sulfonamide

Purity: ≥99%

Product Details
Citations (5)
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Biological Activity

Highly selective muscarinic M1 antagonist (Ki = 14.87 nM). Targets the M1 orthosteric site with greater than 75-fold selectivity over the other receptor subtypes. Reduces pilocarpine-induced seizures in mice. Brain penetrant.

Technical Data

M.Wt:
432.52
Formula:
C18H20N6O3S2
Solubility:
Soluble to 20 mM in DMSO
Purity:
≥99%
Storage:
Store at -20°C
CAS No:
1135243-19-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis. All Tocris products are intended for laboratory research use only.

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Citations for VU 0255035

The citations listed below are publications that use Tocris products. Selected citations for VU 0255035 include:

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